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HuagongsheHuagongshe Chemistry Print Report · For research reference only
HRID 1872254Generated: October 31, 2026

3-Acetoxymethyl-1-(4-methoxy-benzenesulfonyl)-azepane-2-carboxylic acid → 3-Benzofuran-2-yl-1-(4-methoxy-benzenesulfonyl)-2,3,4,7-tetrahydro-1H-azepine-2-carboxylic acid

https://huagongshe.com/reaction/1872254

Reaction equation

Participants

RoleNameHCIDCharge
Reactant3-Acetoxymethyl-1-(4-methoxy-benzenesulfonyl)-azepane-2-carboxylic acidHCID 18689641—
Reactant3-Benzofuran-2-yl-1-(4-methoxy-benzene sulfonyl)-2,3,4,7-tetrahydro-1H-azepine-2-carboxylic acid tert-butyl esterHCID 54397069—
Product3-Benzofuran-2-yl-1-(4-methoxy-benzenesulfonyl)-2,3,4,7-tetrahydro-1H-azepine-2-carboxylic acidHCID 18689669—

Reaction Steps

3-Benzofuran-2-yl-1-(4-methoxy-benzenesulfonyl)-2,3,4,7-tetrahydro-1H-azepine-2-carboxylic acid was synthesized from 3-Benzofuran-2-yl-1-(4-methoxy-benzenesulfonyl)-2,3,4,7-tetrahydro-1H-azepine-2-carboxylic acid tert-butyl ester in the same manner as the procedures used for the preparation of 3-Acetoxymethyl-1-(4-methoxy-benzenesulfonyl)-azepane-2-carboxylic acid: MS (M-H)30 426.

Provenance & Evidence

DOI10.6084/m9.figshare.5104873.v1
Patent numberUS06107291
Source datasetuspto-grants-2000_08
ORD IDord-0e37916ca168463d98f8eff0d380bc63
Source noteuspto-grants-2000_08