HuagongsheHuagongshe Chemistry Print Report · For research reference only
Methyl 4-[5-(cyclopentyloxycarbonyl)amino-1-methylindazol-3-ylmethyl]-3-methoxybenzoate → 4-[5-(Cyclopentyloxycarbonyl)amino-1-methylindazol-3-ylmethyl]-3-methoxybenzoic acid
Participants
| Role | Name | HCID | Charge |
|---|---|---|---|
| Reactant | Methyl 4-[5-(cyclopentyloxycarbonyl)amino-1-methylindazol-3-ylmethyl]-3-methoxybenzoate | HCID 14626827 | — |
| Reactant | 4-[6-(2-ethylhexanamido)indole-1-yl-methyl]-3-methoxybenzoic N,N-diphenylcarbamic anhydride | HCID 14753011 | — |
| Product | 4-[5-(Cyclopentyloxycarbonyl)amino-1-methylindazol-3-ylmethyl]-3-methoxybenzoic acid | HCID 14626829 | — |
Reaction Steps
Using a similar procedure to that described in part (d) of Example 1, except starting from the ester (Y) instead of the ester (C), 4-[5-(cyclopentyloxycarbonyl)amino-1-methylindazol-3-ylmethyl]-3-methoxybenzoic acid (U) was obtained as a white solid (95%); mp 216°-217° C.
Provenance & Evidence
| DOI | 10.6084/m9.figshare.5104873.v1 |
|---|---|
| Patent number | US04837235 |
| Source dataset | uspto-grants-1989_06 |
| ORD ID | ord-c194e3c84251419f9351895cc5cb020f |
| Source note | uspto-grants-1989_06 |