6-Morpholinonicotinic Acid → HCID 178523706, compound

Participants

Reaction Steps

The title compound, white solid (108 mg, 83%), MS (ISP) m/z=521.5 [(M+H)+], mp 222° C., was prepared in accordance with the general method of example 32 from trans-4-{2-[4-(2,3-dihydrofuro[3,2-c]pyridin-4-yl)-piperazin-1-yl]-ethyl}-cyclohexanamine trihydrochloride (intermediate C) (110 mg, 0.25 mmol) and 6-morpholin-4-yl-nicotinic acid.

Provenance & Evidence