HuagongsheHuagongshe Chemistry Print Report · For research reference only
1,2-Oxazole-5-carboxylic acid → HCID 71229238, compound
Participants
| Role | Name | HCID | Charge |
|---|---|---|---|
| Reactant | 1,2-Oxazole-5-carboxylic acid | HCID 2060599 | — |
| Reactant | HCID 60141184 | HCID 60141184 | — |
| Product | HCID 71229238 | HCID 71229238 | — |
Reaction Steps
In analogy to the procedures described for the preparation of intermediate A-1 [B], 1-amino-cyclopropanecarboxylic acid{(rac)-3-[5-chloro-3-fluoro-2-(2-methyl-2H-tetrazol-5-yl)-phenyl]-6,7-dihydro-5H-[1]pyrindin-7-yl}-amide (example 55) was coupled with isoxazole-5-carboxylic acid to yield the title compound as light yellow solid. MS: 523.1 (MH+, 1Cl).
Provenance & Evidence
| DOI | 10.6084/m9.figshare.5104873.v1 |
|---|---|
| Patent number | US08592426B2 |
| Source dataset | uspto-grants-2013_11 |
| ORD ID | ord-dc8ac1245bb54198b1da9a1f334e08c9 |
| Source note | uspto-grants-2013_11 |