2-Butanamine, 2-methyl- → HCID 14988385, compound

Participants

Reaction Steps

A solution of 250 mg (1.54 mmol) of (R)-2-(tetrazolo[1,5-a]pyrid-6-yl)oxirane and 663 mg (7.61 mmol) of tert amylamine in 0.6 ml of absolute ethanol in a pressure tube was heated at 100° C. (bath temperature) for two hours. The reaction mixture was concentrated under reduced pressure to yield 369 mg of crude product which was used in the next reaction without further purification.

Provenance & Evidence