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HuagongsheHuagongshe Chemistry Print Report · For research reference only
HRID 2075213Generated: November 1, 2026

Methyl 1-(3-bromobenzyl)azetidine-3-carboxylate → Methyl 1-(3-(5-benzylbenzofuran-2-yl)benzyl)azetidine-3-carboxylate

https://huagongshe.com/reaction/2075213

Reaction equation

Participants

RoleNameHCIDCharge
ReactantMethyl 1-(3-bromobenzyl)azetidine-3-carboxylateHCID 58415353—
ReactantHCID 59595866HCID 59595866—
ProductMethyl 1-(3-(5-benzylbenzofuran-2-yl)benzyl)azetidine-3-carboxylateHCID 58415396—

Reaction Steps

Synthesized according to Scheme B2, Step 2 and general procedure F from 5-benzylbenzofuran-2-ylboronic acid and methyl 1-(3-bromobenzyl)azetidine-3-carboxylate to give methyl 1-(3-(5-benzylbenzofuran-2-yl)benzyl)azetidine-3-carboxylate as a light yellow oil. MS (ESI) m/z: Calculated: 411.2; Observed: 412 (M++1).

Provenance & Evidence

DOI10.6084/m9.figshare.5104873.v1
Patent numberUS07919519B2
Source datasetuspto-grants-2011_04
ORD IDord-920d40db4a5241aeb6e4b4fe8809131f
Source noteuspto-grants-2011_04