Ethyl 3-{[(4-aminophenyl)carbonyl](methyl)amino}propanoate → 3-[({4-[(1-{1-ethyl-3-[4-(trifluoromethoxy)phenyl]-1H-pyrazol-5-yl}-3-methylbutyl)amino]phenyl}carbonyl)(methyl)amino]propanoic acid

Participants

Reaction Steps

Using 1-{1-ethyl-3-[4-(trifluoromethoxy)phenyl]-1H-pyrazol-5-yl}-3-methylbutan-1-ol (0.39 g) synthesized above and ethyl 3-{[(4-aminophenyl)carbonyl](methyl)amino}propanoate (0.28 g) synthesized in Example 2(2) and in the same manner as in Example 1(7), the title object compound (0.02 g, 4%) was obtained as a white solid.

Provenance & Evidence