HuagongsheHuagongshe Chemistry Print Report · For research reference only
tert-Butyl 2-(aminomethyl)morpholine-4-carboxylate → tert-Butyl 2-({[4-(5-cyano-7-isopropyl-1,3-benzoxazol-2-yl)benzoyl]amino}methyl)morpholine-4-carboxylate
Participants
| Role | Name | HCID | Charge |
|---|---|---|---|
| Reactant | tert-Butyl 2-(aminomethyl)morpholine-4-carboxylate | HCID 19081094 | — |
| Reactant | 4-(5-Cyano-7-isopropylbenzo[d]oxazol-2-yl)benzoic acid | HCID 57369945 | — |
| Product | tert-Butyl 2-({[4-(5-cyano-7-isopropyl-1,3-benzoxazol-2-yl)benzoyl]amino}methyl)morpholine-4-carboxylate | HCID 59586039 | — |
Reaction Steps
The title compound was then prepared from tert-butyl 2-(aminomethyl)morpholine-4-carboxylate (48 mg) and 4-(5-cyano-7-isopropyl-1,3-benzoxazol-2-yl)benzoic acid, INTERMEDIATE 2) as described in EXAMPLE 35. Mass spectrum (ESI) 505.3 (M+1).
Provenance & Evidence
| DOI | 10.6084/m9.figshare.5104873.v1 |
|---|---|
| Patent number | US08445480B2 |
| Source dataset | uspto-grants-2013_05 |
| ORD ID | ord-a854a945614e4bfebd069fca354a5925 |
| Source note | uspto-grants-2013_05 |