Sodium borohydride → HCID 85429906, compound

Participants

Reaction Steps

[(5-{1-[4-(3,3-Dimethyl-2-oxo-butoxy)-3-methyl-phenyl]-1-ethyl-propyl}-benzofuran-2-carbonyl)-methyl-amino]-acetic acid (130 mg, 0.256 mmol) in THF (2.0 mL) are reacted with NaBH4 (19 mg, 0.513 mmol) analogous to Example 8 to yield title compound (120 mg, 92%). MS (ES) m/e: 508.3 (M−1), 510.3 (M+1)

Provenance & Evidence