Morpholine → HCID 68905004, compound

Participants

Reaction Steps

In an analogous manner to EXAMPLE 1, step 3 (1RS,2SR)-1-(1H-indol-1-yl)-3-(4-methylpiperazin-1-yl)-1-phenylpropan-2-ol hydrochloride was prepared from (2RS,3RS)-toluene-4-sulfonic acid 2-hydroxy-3-indol-1-yl-3-phenyl-propyl ester (EXAMPLE 1, step 3) and morpholine. MS (ESI) m/z 337 ([M+H]+); HRMS: calcd for C21H24N2O2+H+, 337.19105; found (ESI, [M+H]+), 337.1909.

Provenance & Evidence