HuagongsheHuagongshe Chemistry Print Report · For research reference only
Furan-3-boronic acid → Methyl 3-(furan-3-yl)-2-methoxy-6-(piperidin-1-ylsulphonylmethyl)benzoate
Participants
| Role | Name | HCID | Charge |
|---|---|---|---|
| Reactant | Furan-3-boronic acid | HCID 2734358 | — |
| Reactant | Ethyl 6-benzenesulphonylmethyl-3-(furan-3-yl)-2-hydroxybenzoate | HCID 67107629 | — |
| Reactant | HCID 69915004 | HCID 69915004 | — |
| Product | Methyl 3-(furan-3-yl)-2-methoxy-6-(piperidin-1-ylsulphonylmethyl)benzoate | HCID 69915016 | — |
Reaction Steps
Prepared by proceeding in a similar manner to Intermediate 36, starting from methyl 3-bromo-2-methoxy-6-(piperidin-1-ylsulphonylmethyl)benzoate (Intermediate 147) and furan-3-boronic acid as a white solid.
Provenance & Evidence
| DOI | 10.6084/m9.figshare.5104873.v1 |
|---|---|
| Patent number | US09067905B2 |
| Source dataset | uspto-grants-2015_06 |
| ORD ID | ord-8846804073a14d55a89eec33c97d6185 |
| Source note | uspto-grants-2015_06 |