HRID2202478

反应详情

EQUATION

反应方程式

HRID 2202478 的结构方程式

PROCEDURE

实验过程

The title compound, white solid (12 mg, 14%), MS (ISP) m/z=433.4 [(M+H)+], mp 247° C., was prepared in accordance with the general method of example 1 from 6-bromo-1-(4-methylsulfonyl-phenyl)-1H-benzo[d]imidazole (intermediate O) (70 mg, 199 μmol) and 1-(4-fluoro-phenyl)-1H-pyrazol-5-ylboronic acid (intermediate A) (49.2 mg, 239 μmol).