2-(5-Bromopentyl)-1H-1lambda~6~,2-benzothiazole-1,1,3(2H)-trione → HCID 131719169, compound

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Reaction Steps

This compound was prepared analogous to the method described for 2-(4-(4-(7-bromo-2,3-dihydro-1,4-benzodioxin-5-yl)-1-piperazinyl)-butyl)-1,2-benzisothiazole-3(2H)-one-1,1-dioxide, dihydrochloride (Example 3) using intermediate 2a (2.00 g, 6.9 mmol) and 2(5-bromopentyl)-1,2-benzisothiazole-3(2H)-one-1,1-dioxide (2.52 g, 7.6 mmol). Yield 1.40 g, m.p. 193°-5° C.

Provenance & Evidence