HuagongsheHuagongshe Chemistry Print Report · For research reference only
Boc-D-phe-pro-OH → Tert-butyl (1r)-1-benzyl-2-oxo-2-{(2s)-2-[(4,5,6,7-tetrahydro-2h-indazol-5-ylamino)carbonyl]pyrrolidinyl}ethylcarbamate
Participants
| Role | Name | HCID | Charge |
|---|---|---|---|
| Reactant | Boc-D-phe-pro-OH | HCID 1797945 | — |
| Reactant | 4,5,6,7-tetrahydro-1H-indazol-5-amine dihydrochloride | HCID 178478653 | — |
| Product | Tert-butyl (1r)-1-benzyl-2-oxo-2-{(2s)-2-[(4,5,6,7-tetrahydro-2h-indazol-5-ylamino)carbonyl]pyrrolidinyl}ethylcarbamate | HCID 178454148 | 80% |
Reaction Steps
The title compound was prepared from Boc-D-PheL-Pro-OH and 5-amino-4,5,6,7-tetrahydro-2H-indazole dihydrochloride using the procedure of EXAMPLE 6, and was obtained as a white solid.
Provenance & Evidence
| DOI | 10.6084/m9.figshare.5104873.v1 |
|---|---|
| Patent number | US07112590B2 |
| Source dataset | uspto-grants-2006_09 |
| ORD ID | ord-b1fb6d9cdfde4cfdb0f53dbe65797b0b |
| Source note | uspto-grants-2006_09 |