HCID 69287896, compound → HCID 11203184, compound

Participants

Reaction Steps

According to the procedure described fort he synthesis of Example 96 further derivatives have been synthesised from 2-[(4-Chloro-phenyl)-(2,4-dichloro-benzoyl)-amino]-5-methyl-thiazole-4-carboxylic acid or 2-[(2,4-Dichloro-benzoyl)-(3,4-dimethoxy-phenyl)-amino]-5-methyl-thiazole-4-carboxylic acid and various commercially available amines and comprise Examples 97-Example 124 below. In cases of Example 102 and 118 additionally 2 eq. NEt3 were added to the reaction mixture as amine hydrochlorides were used as starting materials.

Provenance & Evidence