Pyrrolidine → HCID 10409792, compound

HRID 222686Notes

Reaction equation

HRID 222686 reaction equation
[NH:1]1[CH2:5][CH2:4][CH2:3][CH2:2]1.[CH:6]1([N:11]2[CH2:17][CH2:16][C:15]3[CH:18]=[C:19]([O:22][CH2:23][C:24]4[CH:25]=[C:26]([CH:30]=[CH:31][CH:32]=4)[C:27](O)=[O:28])[CH:20]=[CH:21][C:14]=3[CH2:13][CH2:12]2)[CH2:10][CH2:9][CH2:8][CH2:7]1>>[CH:6]1([N:11]2[CH2:17][CH2:16][C:15]3[CH:18]=[C:19]([O:22][CH2:23][C:24]4[CH:25]=[C:26]([C:27]([N:1]5[CH2:5][CH2:4][CH2:3][CH2:2]5)=[O:28])[CH:30]=[CH:31][CH:32]=4)[CH:20]=[CH:21][C:14]=3[CH2:13][CH2:12]2)[CH2:7][CH2:8][CH2:9][CH2:10]1

Participants

3

Reactant 2

HCID 31268PyrrolidineHCID 10338863HCID 10338863, compound

Product 1

HCID 10409792HCID 10409792, compound

Procedure

Example 96 (E96) was prepared from pyrrolidine and 3-(3-cyclopentyl-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-yloxymethyl)-benzoic acid (E95) using the procedure outlined for Example 90 (E90); MS (ES+), m/e 419 [M+H]+.

Sources & evidence

ORD record
ord-2c9b1def8b8040b4b6e80d5dac72428d
Source dataset
uspto-grants-2012_06
Patent number
US08207331B2

Reaction notes

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