Phenylboronic Acid → HCID 135961881, compound

HRID 2234135Notes

Reaction equation

HRID 2234135 reaction equation
[NH:1]1[C:9]2[C:4](=[CH:5][CH:6]=[CH:7][CH:8]=2)[CH:3]=[C:2]1[C:10]1[C:11](=[O:24])[NH:12][N:13]=[C:14]([C:16]2[CH:17]=[N:18][C:19]([O:22]C)=[CH:20][CH:21]=2)[CH:15]=1.[C:25]1(B(O)O)[CH:30]=[CH:29][CH:28]=[CH:27][CH:26]=1>>[O:22]=[C:19]1[NH:18][CH:17]=[C:16]([C:14]2[CH:15]=[C:10]([C:2]3[NH:1][C:9]4[C:4]([C:3]=3[C:25]3[CH:30]=[CH:29][CH:28]=[CH:27][CH:26]=3)=[CH:5][CH:6]=[CH:7][CH:8]=4)[C:11](=[O:24])[NH:12][N:13]=2)[CH:21]=[CH:20]1

Participants

3

Reactant 2

HCID 66827Phenylboronic AcidHCID 135961866HCID 135961866, compound

Product 1

HCID 135961881HCID 135961881, compound

Procedure

This compound is synthesized, starting from 4-(1H-Indol-2-yl)-6-(6-methoxy-pyridin-3-yl)-2H-pyridazin-3-one, and using phenyl boronic acid, analogously to example 173. Yield 30 mg. LC-MS (ES+) 381 (M+H)+.

Workup

  1. customThis compound is synthesized

Sources & evidence

ORD record
ord-6f3206c687c24043b880126958252f90
Source dataset
uspto-grants-2010_05
Patent number
US07709466B2

Reaction notes

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