4-Toluenesulfonyl chloride → HCID 24825931, compound

HRID 2242068Notes

Reaction equation

HRID 2242068 reaction equation
[C:1]1([CH3:11])[CH:6]=[CH:5][C:4]([S:7](Cl)(=[O:9])=[O:8])=[CH:3][CH:2]=1.[Cl:12][C:13]1[CH:14]=[N:15][CH:16]=[C:17]([Cl:41])[C:18]=1/[CH:19]=[C:20](\[O:31][C:32](=[O:40])[C:33]1[CH:38]=[CH:37][C:36]([NH2:39])=[CH:35][CH:34]=1)/[C:21]1[CH:26]=[CH:25][C:24]([O:27][CH3:28])=[C:23]([O:29][CH3:30])[CH:22]=1>>[C:1]1([CH3:11])[CH:6]=[CH:5][C:4]([S:7]([NH:39][C:36]2[CH:37]=[CH:38][C:33]([C:32]([O:31]/[C:20](/[C:21]3[CH:26]=[CH:25][C:24]([O:27][CH3:28])=[C:23]([O:29][CH3:30])[CH:22]=3)=[CH:19]\[C:18]3[C:17]([Cl:41])=[CH:16][N:15]=[CH:14][C:13]=3[Cl:12])=[O:40])=[CH:34][CH:35]=2)(=[O:9])=[O:8])=[CH:3][CH:2]=1

Participants

3

Reactant 2

HCID 73974-Toluenesulfonyl chlorideHCID 24825928HCID 24825928, compound

Product 1

HCID 24825931HCID 24825931, compound

Procedure

The compound was obtained starting from 4-toluenesulfonyl chloride and 4-amino -benzoic acid (Z)-2-(3,5-dichloro-pyridin-4-yl)-1-(3,4-dimethoxy -phenyl)vinyl ester, following the procedure of Example 16.

Workup

  1. customThe compound was obtained

Sources & evidence

ORD record
ord-cab8c7eb66404f019fa787fdabfb7a60
Source dataset
uspto-grants-2010_03
Patent number
US07671066B2

Reaction notes

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