4-Aminotetrahydropyran → HCID 59639536, compound

Participants

Reaction Steps

Following the general procedure outlined in Example 126, the product of Example 121(150 mg, 0.35 mmol), and 4-aminotetrahydropyran (179 mg, 1.77 mmol) were reacted to give the crude material, which was purified as described in Example 198 to give the desired product 140 mg (90%). LC-MS: 445.4 (MH+, m/z), 2.27 (Rt, min).

Provenance & Evidence