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HuagongsheHuagongshe Chemistry Print Report · For research reference only
HRID 2251133Generated: November 2, 2026

4-(Tetrahydro-2H-pyran-2-yloxy)phenylboronic Acid (contains varying amounts of Anhydride) → 8-[4-(Tetrahydro-pyran-2-yloxy)-phenyl]-5H,7H-6-oxa-1,4,8a-triaza-s-indacene

https://huagongshe.com/reaction/2251133

Reaction equation

Participants

RoleNameHCIDCharge
Reactant4-(Tetrahydro-2H-pyran-2-yloxy)phenylboronic Acid (contains varying amounts of Anhydride)HCID 5017652—
Reactant10-(4-benzyloxy-phenyl)-6,7,8,9-tetrahydro-5H-1,4,10a-triaza-cyclohepta[f]indeneHCID 58587717—
Reactant8-Chloro-5H,7H-6-oxa-1,4,8a-triaza-s-indaceneHCID 58587718—
Product8-[4-(Tetrahydro-pyran-2-yloxy)-phenyl]-5H,7H-6-oxa-1,4,8a-triaza-s-indaceneHCID 58587723—

Reaction Steps

Using the method described for the preparation of 10-(4-benzyloxy-phenyl)-6,7,8,9-tetrahydro-5H-1,4,10a-triaza-cyclohepta[f]indene, the reaction of 8-Chloro-5H,7H-6-oxa-1,4,8a-triaza-s-indacene and 4-(Tetrahydro-pyran-2-yloxy)-phenyl boronic acid provided the title compound.

Provenance & Evidence

DOI10.6084/m9.figshare.5104873.v1
Patent numberUS07319103B2
Source datasetuspto-grants-2008_01
ORD IDord-1186467dfa98428fa6dbb2cf88e10fde
Source noteuspto-grants-2008_01