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HuagongsheHuagongshe Chemistry Print Report · For research reference only
HRID 2276917Generated: October 25, 2026

Potassium trifluoro[(pyrrolidin-1-yl)methyl]borate → 1-[4-(7-Fluoro-2,3-dihydro-benzo[1,4]dioxin-2-yl)-benzyl]-pyrrolidine

https://huagongshe.com/reaction/2276917

Reaction equation

Participants

RoleNameHCIDCharge
ReactantPotassium trifluoro[(pyrrolidin-1-yl)methyl]borateHCID 45588176—
ReactantHCID 68292423HCID 68292423—
Product1-[4-(7-Fluoro-2,3-dihydro-benzo[1,4]dioxin-2-yl)-benzyl]-pyrrolidineHCID 68292691—

Reaction Steps

The title compound is prepared from G-4 and Potassium 1-trifluoroboratomethylpyrrolidine according to the procedure described for the synthesis of compound 202. 203: LC/MS Method 10; Rt=1.07 min.; [M+H]+=354.4.

Provenance & Evidence

DOI10.6084/m9.figshare.5104873.v1
Patent numberUS09133146B2
Source datasetuspto-grants-2015_09
ORD IDord-4ea7a01a7dc34a4e91e7b4bf66c76cbb
Source noteuspto-grants-2015_09