Benzenamine, 4-(4-morpholinyl)- → HCID 178514686, compound

HRID 2284248Notes

Reaction equation

HRID 2284248 reaction equation
[O:1]1[CH2:6][CH2:5][N:4]([C:7]2[CH:13]=[CH:12][C:10]([NH2:11])=[CH:9][CH:8]=2)[CH2:3][CH2:2]1.[NH2:14][S:15]([C:18]1[CH:35]=[CH:34][C:21]2[NH:22][C:23]([C:25]3[CH:33]=[CH:32][C:28]([C:29]([O-])=[O:30])=[CH:27][CH:26]=3)=[N:24][C:20]=2[CH:19]=1)(=[O:17])=[O:16]>>[NH2:14][S:15]([C:18]1[CH:35]=[CH:34][C:21]2[NH:22][C:23]([C:25]3[CH:26]=[CH:27][C:28]([C:29]([NH:11][C:10]4[CH:12]=[CH:13][C:7]([N:4]5[CH2:3][CH2:2][O:1][CH2:6][CH2:5]5)=[CH:8][CH:9]=4)=[O:30])=[CH:32][CH:33]=3)=[N:24][C:20]=2[CH:19]=1)(=[O:16])=[O:17]

Participants

3

Reactant 2

HCID 75655Benzenamine, 4-(4-morpholinyl)-HCID 178514687HCID 178514687, compound

Product 1

HCID 178514686HCID 178514686, compound

Procedure

Compound 482 was prepared from 4-morpholinoaniline and 4-(5-aminosulfonyl-1H-benzimidazol-2-yl)benzoate by standard conditions. [M+H]+ calcd for C24H23N5O4S: 478.16; found: 477.93.

Sources & evidence

ORD record
ord-429e5a581b154bd0a829acf93cc04cab
Source dataset
uspto-grants-2015_09
Patent number
US09144557B2

Reaction notes

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