tert-Butyl bromoacetate → HCID 67687710, compound

Participants

Reaction Steps

Compound 987 was prepared according to the procedure described in Scheme IV from 5-amino-1-(4-aminophenyl)indazole, t-butyl bromoacetate, and 4-morpholinobenzoic acid. 1H NMR (500 MHz, CDCl3) δ 8.15 (s, 1H), 8.09 (s, 1H), 7.98 (s, 1H), 7.84 (d, J=7.5 Hz, 2H), 7.55 (d, J=9 Hz, 1H), 7.48 (d, J=10 Hz, 1H), 7.46 (d, J=7 Hz, 2H), 7.26 (s, 1H), 6.90 (d, J=7.5 Hz, 2H), 6.71 (d, J=7 Hz. 2H), 4.45 (s, 1H), 3.87-3.83 (m, 6H), 3.27-3.25 (m, 4H), 1.51 (m, 9H).

Provenance & Evidence