HCID 15126588, compound → HCID 86751657, compound

Participants

Reaction Steps

In an analogous manner to that described in Example 23, by condensing N-[(S)-α-[(tert-butylsulphonyl)methyl]hydrocinnamoyl]-1-(2,4-dinitrophenyl)-L-histidine and (2R,3S)-3-amino-4-cyclohexyl-1-cyclopropyl-2-hydroxy-1-butanone there is obtained (S)-α-[(S)-α-(tert-butylsulphonyl)methyl]hydrocinnamamido]-N-[(1S,2R)-1-(cyclohexylmethyl)-3-cyclopropyl-2-hydroxy-3-oxopropyl]-1-(2,4-dinitrophenyl)imidazole-4-propionamide as a yellow solid, MS: 795 (M+H)+.

Provenance & Evidence