4-(Methylthio)phenylboronic acid → HCID 18376028, compound

Participants

Reaction Steps

By using 3-bromo-2-(4-fluorophenyl)pyrazolo[1,5-a]pyridine (4.0 g, 13.8 mmol) and 4-methylsulphanyl-phenylboronic acid (3.07 g, 1.83 mmol) the title compound was obtained as a white solid (2.29 g 50%) in the manner described in Example 2. MH+: 335; NMR: (CDCl3) δ 2.53 (3H, s) 6.80 (1H, t) 7.00 (2H, t) 7.15 (1H, t) 7.25 (2H, d) 7.30 (1H, d) 7.50 (2H, d) 7.60 (2H, m) 8.50 (1H, d).

Provenance & Evidence