HCID 58816578, compound → HCID 11398024, compound

Participants

Reaction Steps

To a solution of (2-ethyl-6-methyl-pyridin-4-yl)-carbamic acid pentafluorophenyl ester (Example C13., 0.2M, 3 mL, 0.6 mmol) is added a solution of N-[1-(2-amino-ethyl)-piperidin-4-yl]-4-fluoro-N-propyl-benzenesulfonamide (Example B6., 182 mg, 0.53 mmol). The mixture is stirred at r.t. for 15 h. The mixture is evaporated and the residue purified by HPLC to provide the title compound.

Provenance & Evidence