2-Amino-6-chloropyridine → HCID 59437545, compound

Participants

Reaction Steps

The title compound was prepared following procedure described for intermediate A1 step a), but starting from 2-amino-6-chloropyridine (2.05 g; 16.0 mmol; 1.0 eq.) and ethyl 1-(t-butoxycarbonyl)pyrrole-2-boronic acid (5.06 g; 24.0 mmol; 1.5 eq.) as a beige powder (1.15 g, 27%). HPLC, Rt: 2.65 min. (purity 97.0%). LC/MS, M+(ESI): 204.3.

Provenance & Evidence