(4-Methoxyphenyl)boronic acid → HCID 50991729, compound

HRID 240853Notes

Reaction equation

HRID 240853 reaction equation
Br[C:2]1[C:10]2[C:5](=[CH:6][C:7]([C:11]3[CH:16]=[CH:15][CH:14]=[C:13]([N+:17]([O-:19])=[O:18])[CH:12]=3)=[CH:8][CH:9]=2)[N:4]([C:20]2[CH:25]=[CH:24][N:23]=[CH:22][CH:21]=2)[CH:3]=1.[CH3:26][O:27][C:28]1[CH:33]=[CH:32][C:31](B(O)O)=[CH:30][CH:29]=1>>[CH3:26][O:27][C:28]1[CH:33]=[CH:32][C:31]([C:2]2[C:10]3[C:5](=[CH:6][C:7]([C:11]4[CH:16]=[CH:15][CH:14]=[C:13]([N+:17]([O-:19])=[O:18])[CH:12]=4)=[CH:8][CH:9]=3)[N:4]([C:20]3[CH:25]=[CH:24][N:23]=[CH:22][CH:21]=3)[CH:3]=2)=[CH:30][CH:29]=1

Participants

3

Reactant 2

HCID 201262(4-Methoxyphenyl)boronic acidHCID 50991464HCID 50991464, compound

Product 1

HCID 50991729HCID 50991729, compound

Procedure

The target compound was prepared as in Example 13 using 3-bromo-6-(3-nitrophenyl)-1-(pyridin-4-yl)-1H-indole (97 mg, 0.222 mmol) and 4-methoxyphenylboronic acid (37 mg, 0.244 mmol).

Sources & evidence

ORD record
ord-d13f0a862225411e9c7bf4e669bb38e5
Source dataset
uspto-grants-2014_02
Patent number
US08648089B2

Reaction notes

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