4-(4-Fluorophenyl)piperidine → HCID 71178899, compound

Participants

Reaction Steps

Using ethyl 7-(2-chlorophenylamino)-3-[N-(2-methoxyethyl)sulfamoyl]pyrazolo[1,5-a]pyrimidine-6-carboxylate (0.459 g, 1.008 mmol) obtained in step 1 and 4-(4-fluorophenyl)piperidine (0.158 g, 0.881 mmol) instead of 4-phenylpiperidine, and in the same manner as in Example 1 step 4, the title compound (0.086 g, 15%) was obtained.

Provenance & Evidence