HuagongsheHuagongshe Chemistry Print Report · For research reference only
1,3-Propanesultam → HCID 71252531, compound
Participants
| Role | Name | HCID | Charge |
|---|---|---|---|
| Reactant | 1,3-Propanesultam | HCID 642157 | — |
| Reactant | HCID 86676769 | HCID 86676769 | — |
| Product | HCID 71252531 | HCID 71252531 | 66.1% |
Reaction Steps
Using (5-bromopyrazin-2-yl)[4-(5-cyclopropyl-3-methylpyridin-2-yl)piperazin-1-yl]methanone (150 mg) described in Preparation Example 243 and isothiazolidine 1,1-dioxide (54 mg) and by the reaction and treatment in the same manner as in Example 1, the title compound (109 mg) was obtained.
Provenance & Evidence
| DOI | 10.6084/m9.figshare.5104873.v1 |
|---|---|
| Patent number | US08816079B2 |
| Source dataset | uspto-grants-2014_08 |
| ORD ID | ord-0937a83bb8b14c92b0eeb4838c856819 |
| Source note | uspto-grants-2014_08 |