Dimethylamine tetrahydrofuran → HCID 71253196, compound

Participants

Reaction Steps

Using N,N-di-tert-butyloxycarbonyl-2-[4-(5-cyclopropyl-3-methylpyridin-2-yl)piperazine-1-carbonyl]-5-(1,1-dioxo-1λ6-isothiazolidin-2-yl)benzamide (100 mg) described in Example 805 and 2 mol/L dimethylamine tetrahydrofuran solution (88 μL) and by the reaction and treatment in the same manner as in Example 770, the title compound (41 mg) was obtained.

Provenance & Evidence