Anthranilic Acid → HCID 11590082, compound

HRID 2422653Notes

Reaction equation

HRID 2422653 reaction equation
[C:1]([OH:10])(=O)[C:2]1[C:3](=[CH:5][CH:6]=[CH:7][CH:8]=1)[NH2:4].[CH3:11][NH2:12].[CH3:13][C:14]1[CH:21]=[C:20]([O:22][CH3:23])[CH:19]=[CH:18][C:15]=1[CH:16]=O.OC1[CH2:30][CH2:29][N:28](C(OC(C)(C)C)=O)[CH2:27][CH2:26]1.[C:38]1(=O)[CH2:43][CH2:42][CH2:41][CH2:40][CH2:39]1>>[CH3:11][N:12]1[C:1](=[O:10])[C:2]2[C:3](=[CH:5][CH:6]=[CH:7][CH:8]=2)[N:4]=[C:16]1[C:15]1[CH:18]=[CH:19][C:20]([O:22][CH:23]2[CH2:30][CH2:29][N:28]([CH:38]3[CH2:43][CH2:42][CH2:41][CH2:40][CH2:39]3)[CH2:27][CH2:26]2)=[CH:21][C:14]=1[CH3:13]

Participants

6

Reactant 5

HCID 227Anthranilic AcidHCID 6329MethylamineHCID 7967CyclohexanoneHCID 2832854-Methoxy-2-methylbenzaldehydeHCID 643502Tert-butyl 4-hydroxypiperidine-1-carboxylate

Product 1

HCID 11590082HCID 11590082, compound

Procedure

The entitled compound was obtained according to the method of Example 85 but using anthranilic acid, methylamine, 2-methyl-4-methoxybenzaldehyde, tert-butyl 4-hydroxytetrahydro-1(2H)-pyridinecarboxylate, and cyclohexanone.

Workup

  1. customThe entitled compound was obtained

Sources & evidence

ORD record
ord-34a465ee5c8a4dd082901b616ccd0b39
Source dataset
uspto-grants-2011_06
Patent number
US07960394B2

Reaction notes

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