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HuagongsheHuagongshe Chemistry Print Report · For research reference only
HRID 268774Generated: October 30, 2026

(4-Methoxyphenyl)boronic acid → 3-(1H-Indol-6-yl)-3-(4-methoxy-phenyl)-propionic acid methyl ester

https://huagongshe.com/reaction/268774

Reaction equation

Participants

RoleNameHCIDCharge
Reactant(4-Methoxyphenyl)boronic acidHCID 201262—
ReactantHCID 59831848HCID 59831848—
Product3-(1H-Indol-6-yl)-3-(4-methoxy-phenyl)-propionic acid methyl esterHCID 5983161166%

Reaction Steps

3-(1H-Indol-6-yl)-3-(4-methoxy-phenyl)-propionic acid methyl ester XXXIV (0.51 g, 66% yield) was prepared from 4-methoxy boronic acid using the procedure described for preparation of 3-(1H-indol-6-yl)-3-(3-methoxy-phenyl)-propionic acid methyl ester XXXI (see Example 7).

Provenance & Evidence

DOI10.6084/m9.figshare.5104873.v1
Patent numberUS07446118B2
Source datasetuspto-grants-2008_11
ORD IDord-cb4a7514948740aa86727a264170c5a2
Source noteuspto-grants-2008_11