HRID28819

反应详情

EQUATION

反应方程式

HRID 28819 的结构方程式

PROCEDURE

实验过程

In an analogous manner to Example 135, step 3 1-[2-(4-aminopiperidin-1-yl)-1-(3′,4′-dichloro-1,1′-biphenyl-3-ylethyl]cyclohexanol dihydrochloride was prepared from tert-butyl {1-[2-(3′,4′-dichloro-1,1′-biphenyl-3-yl)-2-(1-hydroxycyclohexyl)ethyl]piperidin-4-yl}carbamate. MS (ES) m/z 447.2 ([M+H]+); HRMS: calcd for C25H32Cl2N2O.2.00 HCl, 518.1425; found (ESI), 447.1962.