HRID331414
反应详情
EQUATION
反应方程式
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反应物
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生成物
PROCEDURE
实验过程
The title compound, off-white solid (81 mg, 62%), MS (ISP) m/z=455.4 [(M+H)+], mp 165° C., was prepared in accordance with the general method of example 1 from trans-4-[2-(4-benzofuran-4-yl-piperidin-1-yl)-ethyl]-cyclohexyl-amine dihydrochloride (intermediate A) (115 mg, 0.29 mmol) and rac-(1,4-dioxan-2-yl)-acetic acid.