3-Methoxypropionic acid → HCID 178495576, compound

Participants

Reaction Steps

The title compound, white solid (60 mg, 56%), MS (ISP) m/z=431.5 [(M+H)+], mp 177° C., was prepared in accordance with the general method of example 1 from trans-4-{2-[4-(7-fluoro-benzofuran-4-yl)-piperidin-1-yl]-ethyl}-cyclohexylamine dihydrochloride (intermediate C) (104 mg, 0.25 mmol) and 3-methoxypropionic acid.

Provenance & Evidence