Formaldehyde → HCID 67312034, compound

Participants

Reaction Steps

Prepared as described in the Amination section using sodium cyanoborohydride (67 mg, 1.06 mmol), 4-amino-N-[4-(6-methoxybenzothiazol-2-yl)-phenyl]-benzamide (80 mg, 0.213 mmol) and paraformaldehyde (64 mg, 2.13 mmol) in AcOH (2 ml) to give the title compound (49 mg, 57%) as colourless needles after recrystallisation from EtOH.

Provenance & Evidence