HuagongsheHuagongshe Chemistry Print Report · For research reference only
(Naphthalen-2-yl)boronic acid → 3-(Naphthalen-2-yl)-1-trityl-1H-pyrazolo[4,3-b]pyridine
Participants
| Role | Name | HCID | Charge |
|---|---|---|---|
| Reactant | (Naphthalen-2-yl)boronic acid | HCID 2734375 | — |
| Reactant | 3-Iodo-1-trityl-1H-pyrazolo[4,3-b]pyridine | HCID 68932363 | — |
| Product | 3-(Naphthalen-2-yl)-1-trityl-1H-pyrazolo[4,3-b]pyridine | HCID 68932700 | 28.7% |
Reaction Steps
By treating 731 mg of 3-iodo-1-trityl-1H-pyrazolo[4,3-b]pyridine obtained by Example 418 and 340 mg of 2-naphthalene boronic acid in the manner as described in Production example 194, 210 mg of the title compound was obtained as a colorless powder.
Provenance & Evidence
| DOI | 10.6084/m9.figshare.5104873.v1 |
|---|---|
| Patent number | US07429609B2 |
| Source dataset | uspto-grants-2008_09 |
| ORD ID | ord-fe5376172d2748c08c3fccc8b5ac8ca6 |
| Source note | uspto-grants-2008_09 |