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HuagongsheHuagongshe Chemistry Print Report · For research reference only
HRID 344315Generated: November 3, 2026

Phenylacetyl chloride → HCID 54309550, compound

https://huagongshe.com/reaction/344315

Reaction equation

Participants

RoleNameHCIDCharge
ReactantPhenylacetyl chlorideHCID 7679—
Reactant4-Amino-5-chloro-2-methoxybenzoic acidHCID 81626—
ReactantHCID 53780050HCID 53780050—
ProductHCID 54309550HCID 54309550—

Reaction Steps

4-((3R)-3-tert-Butoxycarbonylaminomethylpyrrolidin-1-yl)butylamine (1.00 g) as starting compound was reacted and treated in the same manner as in Example 1 using phenylacetyl chloride (0.50 ml) and 4-amino-5-chloro-2-methoxybenzoic acid (0.54 g) to give 4-amino-5-chloro-2-methoxy-N-((3R)-1-(4-phenylacetylaminobutyl)pyrrolidin-3-ylmethyl)benzamide.

Provenance & Evidence

DOI10.6084/m9.figshare.5104873.v1
Patent numberUS05864039
Source datasetuspto-grants-1999_01
ORD IDord-badce00865e2477ea8a4aea27bedefa5
Source noteuspto-grants-1999_01