Propyl isocyanate → HCID 53757672, compound

Participants

Reaction Steps

4-((3R)-3 -tert-Butoxycarbonylaminomethylpyrrolidin-1-yl)butylamine (2.00 g) as starting compound was reacted and treated in the same manner as in Example 34 using n-propyl isocyanate (0.76 ml) and 4-amino-5-chloro-2-methoxybenzoic acid (1.49 g) to give 4-amino-5-chloro-2-methoxy-N-((3R)-1-(4-(3-n-propylureido)butyl)pyrrolidin-3-ylmethyl)benzamide.

Provenance & Evidence