Butyl isocyanate → HCID 54298237, compound

Participants

Reaction Steps

5-((3R)-3-tert-Butoxycarbonylaminomethylpyrrolidin-1-yl)pentylamine (2.00 g) as starting compound was reacted and treated in the same manner as in Example 34 using n-butyl isocyanate (0.79 ml) and 4-amino-5-chloro-2-methoxybenzoic acid (0.54 g) to give 4-amino-N-((3R)-1-(5-(3-n-butylureido)pentyl)pyrrolidin-3-ylmethyl)-5-chloro-2-methoxybenzamide.

Provenance & Evidence