4-Amino-5-chloro-2-methoxybenzoic acid → HCID 53649457, compound

Participants

Reaction Steps

2-(2-(3-tert-Butoxycarbonylaminomethylpyrrolidin-1-yl)ethyl)-2,3-dihydro-1 H-isoindole-1,3-dione (1.5 g) as starting compound was reacted and treated in the same manner as in Example 67 using 4-amino-5-chloro-2-methoxybenzoic acid (0.81 g) to give 4-amino-5-chloro-N-(1-(2-(-2,3-dihydro-1 ,3-dioxo-1 H-isoindol-2-yl)ethyl)pyrrolidin-3-ylmethyl)-2-methoxybenzamide.

Provenance & Evidence