HCID 54247374, compound → HCID 54190377, compound

Participants

Reaction Steps

4-Amino-5-chloro-2-methoxy-N-(piperidin-4-ylmethyl)benzamide dihydrochloride (0.98 g) as starting compound and 7-bromo-1-(1-methyl-1 H-indol-3-yl)-1-heptanone were reacted and treated in the same manner as in Example 172 to give 0.83 g of 4-amino-5-chloro-2-methoxy-N-((1-(7-(1-methyl-1 H-indol-3-yl)-7-oxoheptyl)piperidin-4-yl)methyl)-benzamide. This compound was treated with hydrochloric acid-ethanol to obtain its hydrochloride as crystals.

Provenance & Evidence