Acetaldehyde → HCID 69036129, compound

Participants

Reaction Steps

Following the procedure of Example 104 but substituting acetaldehyde for aqueous formaldehyde, 1-([(1S, 2R, 4R)-2-benzenesulfonylmethyl-4-isopropylamino-cyclohexyl)-4-(3-trifluoromethylphenyl)-5,6-dihydro-1H-pyridin-2-one (43 mg, 0.08 mmol) was converted to the title product (45 mg) as a white glassy solid. MS found: (M+H)+=563.29.

Provenance & Evidence