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HuagongsheHuagongshe Chemistry Print Report · For research reference only
HRID 352732Generated: October 25, 2026

4-(Diethylboranyl)pyridine → 1-[2-tert-Butoxycarbonyl-4-(pyridin-4-yl)benzoyl]-4-[(6-chloronaphthalen-2-yl)sulfonyl]piperazine hydrochloride

https://huagongshe.com/reaction/352732

Reaction equation

Participants

RoleNameHCIDCharge
Reactant4-(Diethylboranyl)pyridineHCID 13318871—
Reactant1-[4-Bromo-2-(tert-butoxycarbonyl)benzoyl]-4-[(6-chloronaphthalen-2-yl)sulfonyl]piperazineHCID 22709864—
Product1-[2-tert-Butoxycarbonyl-4-(pyridin-4-yl)benzoyl]-4-[(6-chloronaphthalen-2-yl)sulfonyl]piperazine hydrochlorideHCID 22710746—

Reaction Steps

In the same manner as in Referential Example 7, a reaction was conducted using 1-[4-bromo-2-(tert-butoxycarbonyl)benzoyl]-4-[(6-chloronaphthalen-2-yl)sulfonyl]piperazine and diethyl(4-pyridyl)borane as starting materials, whereby the title compound was obtained.

Provenance & Evidence

DOI10.6084/m9.figshare.5104873.v1
Patent numberUS06747023B1
Source datasetuspto-grants-2004_06
ORD IDord-39f9d244ff6248faa11c697752b1f847
Source noteuspto-grants-2004_06