Pyrazole → HCID 17508634, compound

HRID 367623Notes

Reaction equation

HRID 367623 reaction equation
N1C=CC=N1.Cl[C:7]1[N:8]=[C:9]([NH:18][CH2:19][C:20]2[CH:25]=[CH:24][C:23]3[O:26][CH2:27][CH2:28][O:29][C:22]=3[CH:21]=2)[C:10]2[C:15]([CH3:16])=[C:14]([CH3:17])[S:13][C:11]=2[N:12]=1>>[CH3:16][C:15]1[C:10]2[C:9]([NH:18][CH2:19][C:20]3[CH:25]=[CH:24][C:23]4[O:26][CH2:27][CH2:28][O:29][C:22]=4[CH:21]=3)=[N:8][CH:7]=[N:12][C:11]=2[S:13][C:14]=1[CH3:17]

Participants

3

Reactant 2

HCID 1048PyrazoleHCID 18460333HCID 18460333, compound

Product 1

HCID 17508634HCID 17508634, compound

Procedure

Following the procedure of Example 97, the reaction of pyrazole with 2-chloro-5,6-dimethyl-4-(3,4-ethylendioxybenzylamino)-thieno-[2,3-d]-pyrimidine gives 2-pyrazol-1-yl)-5,6-dimethyl-4-(3,4-ethylendioxybenzylamino)-thieno-[2,3-d]-pyrimidine.

Sources & evidence

ORD record
ord-e5f5cd30a7c64c6eadbb9c256d2149f9
Source dataset
uspto-grants-2000_10
Patent number
US06133271

Reaction notes

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