2-Fluorobenzoyl chloride → HCID 18360382, compound

Participants

Reaction Steps

An amidation reaction and post-treatment were carried out under the same conditions as in Example 22, using 1.50 g (6.40 mol) of 4-amino-1-(2-fluorobenzyl)-5-imidazole carboxamide which was prepared in the same manner as in Example 113 and 2-fluorobenzoyl chloride instead of benzoyl chloride to obtain 2.21 g of 4-(2-fluorobenzoylamino)-1-(2-fluorobenzyl)-5-imidazolecarboxamide (yield 97%).

Provenance & Evidence