2-Fluorobenzoyl chloride → HCID 18360413, compound

Participants

Reaction Steps

An amidation reaction and post-treatment were carried out following the conditions of Example 22, using 1.00 g (4.06 mmol) of 4-amino-1-(2-phenoxyethyl)-5-imidazolecarboxamide prepared in the same manner as in Example 155 and 2-fluorobenzoyl chloride instead of benzoyl chloride to obtain 1.39 g of 4-(2-fluorobenzoylamino)-1-(2-phenoxyethyl)-5-imidazolecarboxamide (yield 93%).

Provenance & Evidence