1H-Indazol-6-amine → HCID 22646658, compound

Participants

Reaction Conditions

Reaction Steps

A suspension of 4-chloro-6,7-dimethoxyquinoline (200 mg, 0.89 mmol), (prepared as described for the starting material in Example 2), and 6-aminoindazole (131 mg, 0.98 mmol) in DMF (2.5 ml) was heated at 140° C. for 1.5 hours. The solid was collected by filtration, washed with isopropanol and dried under vacuum to give 6,7-dimethoxy-4-(1H-indazol-6-ylamino)quinoline hydrochloride (171 mg, 54%).

Provenance & Evidence