1-(Propan-2-yl)piperidin-4-amine → HCID 66624637, compound

Participants

Reaction Steps

[(S)-1-Benzyloxymethyl-2-(1-isopropyl-piperidin-4-ylsulfamoyl)-ethyl]-carbamic acid benzyl ester was prepared by an analogous procedure as described for example 26 vi) starting from 142 mg (1.0 equiv.) 1-isopropyl-piperidin-4-ylamine and 398 mg (1.0 mmol) ((S)-1-benzyloxymethyl-2-chlorosulfonyl-ethyl)-carbamic acid benzyl ester. The product was obtained in crude form as a light yellow foam. Yield: 217 mg MS (ES+): m/e=504.

Provenance & Evidence